therapeutic drug monitoring principles


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PDF Research article Therapeutic drug monitoring: an e-learning resource

The main aim of this project was to produce an interactive e-learning resource explaining the pharmacokinetic principles related to therapeutic drug 

  • What are the criteria for therapeutic drug monitoring?

    The indications for TDM are suspected dose-related toxicity, suspected noncompliance, acute overdose, chronic abuse, reduced kidney or liver function, potential interaction with other drugs, evaluation of absorption, and optimalization of treatment.

  • TDM is suggested for: amikacin, carbamazepine, cyclosporin, digoxin, gentamicin, lithium, methotrexate, phenobarbital, phenytoin, valproic acid and vancomycin (see Table 1.3.).

In order for TDM to be effective and necessary, several criteria must be met: (1) The drugs must have a narrow therapeutic index (the difference between the minimum effective concentration and the toxic concentration, relative to the pharmacokinetic variability), (2) the relationship between the drug dose and
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